Neuro Lab · DeCure for X

DeCure for Vascular dementia

DeCure's autonomous Neuro AI scientist is researching a drug-repurposing hypothesis for vascular dementia — screening already-approved drugs against its 35-gene Open Targets disease module to publish open-access research. Research is fast; the path to publication is funded in milestone stages.

Disease module35 genesLead labNeuro
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NeuroDOID:8725$DeCureNeuro

The disease map

Disease moduleVascular dementia maps to a 35-gene Open Targets module — the target space DeCure's AI scientist screens approved drugs against.
DeCure.ai methodSignature reversal (LINCS) plus network proximity (STRING) rank already-approved drugs likely to perturb this module — the same engine that produces DeCure.ai's repurposing hypotheses.
Repurposing thesisScreening approved medicines against this disease module, then publishing the evidence for the strongest candidate. Known pharmacology and human exposure data make the first question sharper — they do not establish safety or efficacy in a new indication.

Research record

01
ResearchComing soon
Candidate research + dossier — target rationale, drug-repurposing thesis and evidence pack.proof: Published dossier + on-chain hash
02
ValidationComing soon
In-vitro biological validation at a contract research org (CRO).proof: CRO contract + in-vitro report
03
Peer review & paperComing soon
Peer-reviewed paper published open-access (preprint + journal).proof: DOI + open-access link + on-chain hash

Current lead

No approved-drug candidate for vascular dementia is corroborated in the literature DeepSearch retrieved. Some conditions are managed with non-pharmacological care — a device, surgery or physical therapy — rather than a medicine; that may be the case here, or the literature we found may simply be too sparse yet to support a drug-repurposing angle.

Molecular view

KRIT1 ankyrin repeat containing (KRIT1)KRIT1 is one of the genes genetically linked to this disease in Open Targets — shown as context, not as a drug target we're pursuing: no approved-drug candidate for this disease is yet corroborated in the literature we found.

Loading structure…
helix sheet gnpdrag to rotate · scroll to zoom

RCSB Protein Data Bank · entry 4HDO · 1.67 Å · ligand PHOSPHOAMINOPHOSPHONIC ACID-GUANYLATE ESTER (GNP). Experimental structure, not a prediction.

What the evidence adds up to

Vascular dementia is the second most common dementia type, but no truly effective treatments have emerged. A 2016 review notes that while stroke prevention and treatment have transformed over the last 25 years, with falling stroke incidence in most developed countries and rapid treatments after transient ischaemic attack reducing early recurrent stroke to negligible levels, dementia treatment remains absent. The same review states that evidence for individual vascular risk factor interventions preventing or delaying progression of Alzheimer's disease dementia has so far been disappointing, though falling dementia rates in population studies and improved cognitive function in a multifactorial 'vascular health' randomised trial give some hope.

Small vessel disease is the commonest cause of vascular dementia and a central pathway in stroke and dementia pathogenesis. It causes one-fifth of all strokes, and in up to 45% of the estimated 47.5 million people living with dementia worldwide, small vessel disease is a major contributing or the sole pathology. The 2016 review proposes that the cerebral vascular endothelium and blood–brain barrier become leaky, allowing plasma components into the vessel wall and surrounding tissues, causing secondary damage accompanied by inflammatory cell infiltrates, myelin and axonal damage. This theory is gathering momentum, supported by patient studies and experimental models.

A 2011 paper suggests that in the vast majority of cases, vascular dementia occurs in an already aged brain with cellular and molecular events common to different neurodegenerative diseases, and that cell signalling defects and molecular dyshomeostasis may lead to neuronal malfunction before neuron death. The 2016 review emphasises that most dementias in the elderly are mixed vascular and Alzheimer's disease, and that the expression of cognitive impairment for a given age and burden of Alzheimer's pathology is most strongly influenced by the amount of vascular disease rather than by Alzheimer's pathology stage. A 2023 overview states that since vascular dementia is preventable, studying it clinically is important to improve patient prognosis, but provides no new trial data.

What is still missing is a clear mechanistic understanding that can be translated into effective interventions. The 2016 review highlights that dementia research has been dominated by Alzheimer's disease focused on amyloid plaques and tau, with hundreds of interventions tested in mouse models but only 4% of interventions reporting actual outcomes. It calls for wider thinking, better experimental models that reflect mixed pathologies, and joint work between vascular and dementia researchers rather than parallel duplicative efforts. No drug treatment is mentioned in any of these abstracts.

Evidence

Retrieved by DeepSearch across 234,678,978 indexed works and resolved on OpenAlex — ranked by citations, including the results that did not work.

Journal of Aging Research · 2011 · 37 citations · open access

Neurobiology of Vascular Dementia

AbstractVascular dementia is, in its current conceptual form, a distinct type of dementia with a spectrum of specific clinical and pathophysiological features. However, in a very large majority of cases, these alterations occur in an already aged brain, characterized by a milieu of cellular and molecular events common for different neurodegenerative diseases. The cell signaling defects and molecular dyshomeostasis might lead to neuronal malfunction prior to the death of neurons and the alteration of neuronal networks. In the present paper, we explore some of the molecular mechanisms underlying brain malfunction triggered by cerebrovascular disease and risk factors. We suggest that, in the age of genetic investigation and molecular diagnosis, the concept of vascular dementia needs a new approach.

https://doi.org/10.4061/2011/401604
Clinical Science · 2016 · 5 citations · open access

Small vessels, dementia and chronic diseases–molecular mechanisms and pathophysiology

AbstractThis editorial introduces a special themed issue of Clinical Science on vascular causes of dementia, particularly small vessel disease (SVD), the commonest cause of vascular dementia and a central common pathway in the pathogenesis of stroke and dementia.The themed issue, initiated by the Vascular Experimental Theme of the Dementia Platform UK (DPUK), will include critical reviews on several key topics from experts in the field–these are in progress–but we are also keen to receive proffered reviews and original work addressing molecular and translational topics that aim to unravel the complex and multifactorial processes that contribute to development and clinical expression of human cerebral SVD. It complements a workshop, to be held in January 2017, bringing together researchers in dementia and stroke to discuss the multifactorial mechanisms contributing to neurodegeneration acting around the complex vascular–brain interface, including models, their relevance and ways to ensure reliability.These are interesting times for research in stroke and dementia, and for SVD(s) as central underpinning pathologies. Stroke and dementia both generate astoundingly large health and societal problems. Nearly 17 million people have a first stroke each year worldwide [1], of whom about one-third have died from the stroke by 6 months, one-third are dependent and only one-third can continue living independently. Stroke has been the second commonest cause of death in the world and the commonest cause of dependency in older adults consistently for many decades [2,3], and is a common cause of cognitive decline and dementia [4]. SVD causes one-fifth of all strokes (lacunar ischaemic stroke; many haemorrhagic strokes in older people) [5] and worsens outcomes after stroke [6]. There are estimated to be approximately 47.5 million people in the world living with dementia [7], in up to 45% of whom SVD is a major contributing or the sole pathology [8]. This may be an underestimate since dementia may be under-diagnosed, particularly in low- and middle-income countries where healthcare provision is thinly spread and family support within a familiar environment may allow failing cognition to go undetected. Many governments have now made dementia a priority for research to accelerate development of prevention and treatment, with very large research spends.What are the treatment options? The prevention and treatment of stroke have changed almost beyond recognition in the last 25 years, from nihilism, to becoming one of the most, if not the most, preventable and treatable neurological diseases. Consequently, stroke incidence is falling in most developed countries [9], rapid implementation of medical [10] and surgical treatments after transient ischaemic attack or minor stroke can reduce early recurrent stroke to negligible levels [11], and many more patients remain independent after acute ischaemic stroke thanks to stroke units, thrombolysis and thrombectomy [12,13]. There is now evidence that improved stroke prevention and treatment are leading to parallel reductions in diagnoses of dementia [14].In contrast, although several different causes of dementia are now recognized (Alzheimer's disease, fronto-temporal, Lewy body, vascular), truly effective treatments for dementia have yet to emerge, and, apart from possibly adopting a healthy lifestyle [15] and managing modifiable vascular risk factors such as hypertension (both of which are generally good ideas anyway) [16], little can yet be done to prevent dementia, including once early signs of cognitive impairment are evident [17,18].Dementia research is dominated by Alzheimer's disease which has largely focused on amyloid plaques and tau protein. However, despite decades of research, millions spent, hundreds of interventions tested (e.g. over 300 in the Tg2576 mouse model alone [19]), the lack of effective treatment or prevention has led to calls for wider thinking about Alzheimer's disease pathogenesis [20].It has long been evident that most dementias in the elderly are mixed vascular and Alzheimer's disease [21]. Human studies have shown repeatedly that the expression of cognitive impairment or dementia in life, for a given age and burden of Alzheimer's pathology, is most strongly influenced by the amount of vascular disease rather than by the Braak stage or burden of Alzheimer's disease pathology [21–23]. The recent finding of reductions in incidence of dementia paralleling improvements in stroke prevention and treatment [14,24,25], as well as data modelling exercises [26], appear to provide further evidence for important vascular contributions to dementia.A clear mechanistic understanding is fundamental to the development of effective interventions. In stroke, this was accelerated by the advent of neuroimaging from the late 1980s, which allowed more accurate epidemiology to differentiate haemorrhagic from ischaemic stroke, tracking of brain responses to arterial occlusion and re-opening [27] and encouraged trials of thrombolysis and thrombectomy. Imaging with MRI and positron emission tomography (PET) also provided pathophysiological insights into stages of tissue injury in relation to blood flow in human ischaemic stroke [28]. A similar approach, taking advantage of the range of neuroimaging tools which are now substantially more advanced, has been set out recently for Alzheimer's disease [29]. In stroke, information from neuroimaging in patients has also helped to balance suggestions emerging from experimental models that were simply incorrect, for example that reperfusion worsened ischaemic tissue damage after acute ischaemic stroke [30]. As we know now, reperfusion accelerates recovery [31] and is the basis of acute stroke treatment.In stroke, there is a long-running healthy debate on the balance of information from experimental models compared with human clinical research [32]. This has helped to shape awareness of the strengths and limitations of both approaches and led to improved standards for, and reliability of, experimental studies (e.g. the ARRIVE reporting guidelines, http://www.equator-network.org). Models of cerebral SVD, subcortical ischaemic stroke and monogenic SVDs have been reviewed extensively [33,34], including of vascular dementia and the limitations [35,36]. These have also provided valuable confirmatory mechanistic insights that are hard to obtain in humans.Have dementia models received the same scrutiny? Most research into Alzheimer's disease pathophysiology is performed in rodents, but the rodent brain has proportionately much more grey and much less white matter than the human brain. As the interaction between the two is a fundamental component of human cognition, this must influence model relevance and interpretation in relation to human dementia pathologies. There has been less critical appraisal of Alzheimer's disease models but recent work is revealing [19]. A critical appraisal of transgenic mouse models of Alzheimer's disease identified 427 papers describing 55 transgenic models, n=11 118 animals used in 838 experiments testing 357 interventions: blinding, randomization and sample size estimation were mostly lacking, but of even more concern, the actual outcome of the intervention was described for only 16 of 357 interventions tested (4%) [19]. Studies did not give reasons for not reporting results of the other 341 (96%) interventions, but the information would be important to the field.The wider thinking called upon to advance understanding of Alzheimer's disease pathophysiology and treatment [20] can equally be applied to vascular dementia [37] and small vessel stroke. It has long been assumed that microvascular brain damage is ‘ischaemic’ and due to vessel narrowing from atheroma or spasm [5]. This is partly because the white matter lesions commonly seen on brain magnetic resonance scanning appear ‘white’, similar to the appearance of an acute infarct due to a large blocked artery. Although narrowing of the perforating arterioles does occur, there are also areas of dilation, and occluded arterioles have rarely been found in lacunar ischaemic stroke [38]. Cerebral blood flow (CBF) falls with increasing white matter hyperintensity (WMH) burden in humans, but there are no/little data to indicate a longitudinal association between low CBF and worsening WMH [39]; instead, worsening WMH leads to lower CBF [40]. An alternative hypothesis for SVDs suggests that the cerebral vascular endothelium–the blood–brain barrier (BBB)–becomes more leaky and allows plasma components (and cells) into and through the arteriolar and capillary wall, causing secondary damage in the vessel wall and surrounding tissues [41]. The process is accompanied by inflammatory cell infiltrates in the vessel wall and perivascular tissues, secondary myelin and axonal damage. This theory is now gathering momentum [42–45], is supported by studies in patients ([46–48] and summarized in [49]) and experimental models, both of sporadic [50] and monogenic SVDs [51] and translational genetic studies [52].There is still much to unravel. These topics will be addressed in this themed issue, discussed at the workshop, and we welcome additional proffered papers describing original research and reviews.Considering that a broad consensus may be emerging in the dementia field, and recognizing that multifactorial or mixed dementias are probably more common than pure dementia of any type, it may be more valuable to describe an individual's mixed dementia in terms of the proportion due to Alzheimer's disease or vascular pathology [67], because in turn this may assist in determining patient treatment and management. It may be a more realistic reflection of the messy world of multiple concurrent pathologies that accumulate in later life. In which case, the science of clinical research and laboratory methods, particularly the experimental models, need to reflect this reality.Meantime, in the field of stroke, we can at least do a lot to manage vascular risk factors and, while evidence that individual vascular risk factor interventions prevent or delay progression of Alzheimer's disease dementia has so far been disappointing [8,68,69], the falling dementia rates in population-based studies [14] and improved cognitive function in at risk older individuals using a multifactorial ‘vascular health’ approach in a randomized trial [15], give considerable hope that joint scientific endeavours between vascular and dementia researchers at the highly integrated vascular–brain interface are likely to be effective in reducing the burden of dementia and stroke. This requires researchers in stroke, dementia and vascular biology to work together, benefitting from each other's knowledge, rather than pursuing parallel duplicative work, or, worse, repeating earlier erroneous work, which is the risk of remaining on home ground, however appealing that may be.

https://doi.org/10.1042/cs20160376
Journal of Clinical and Nursing Research · 2023 · 0 citations · open access

Pathogenesis, Rehabilitation Assessment, Treatment Status, and Research Progress of Vascular Dementia

AbstractGiven the global trends in population aging, the prevalence of vascular dementia (VD) is increasing year by year. VD has become the second most common type of dementia and can seriously threaten the quality of life of patients. Since VD is preventable, it is important to study VD clinically in order to improve the prognosis of patients. In recent years, a large number of studies have been carried out at home and abroad, focusing on the pathogenesis, rehabilitation assessment, and treatment of VD. This article is a concise overview of these studies.

https://doi.org/10.26689/jcnr.v7i4.5116
NATIONAL JOURNAL OF NEUROLOGY · 2021 · 0 citations · open access

AbstractThis review article summarizes the information published over the past 10 years on the treatment of noncognitive impairment, which is the most common reason for patients with vascular dementia to seek psychiatric care and hospitalization.Timely treat ment of these symptoms is very important for both the patient and the caregiver.Pathomorphosis in the clinic of vascular dementia has created a need for new methods of treatments.The purpose of this article is to gather uptodate information about treatment of neuropsychiatric symptoms in vascular dementia.We believe that this review article will be one of the steps taken in this direction.

https://doi.org/10.61788/njn.v1i21

Disease module: DeepOracle (Open Targets). Structures: RDKit from PubChem SMILES. Literature: retrieved by DeepSearch across 234,678,978 indexed works (targeted per-candidate search), resolved on OpenAlex.

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